Contents: 1. Introduction to Biopharmaceutics 2. Absorption of Drugs from Gastrointestinal Tract 3. Drug Distribution 4. Drug Elimination 5. Pharmacokinetics: Basic Concepts 6. One Compartment Open Model 7. Multi-Compartment Models 8. Multiple-Dose Regimens 9. Non-linear Pharmacokinetics 10. Non-compartmental Pharmacokinetics 11. Bioavailability and Bioequivalence 12. Biostatistics 13. In-vitro Dissolution Testing